Adrenergic Receptor Inhibitors

α adrenergic receptor

β adrenergic receptor

Adrenergic Receptor Inhibitors, Agonists, Antagonists, Activators, Modulators & Ligands

Product Name	α adrenergic receptor	β adrenergic receptor	Purity
Isoprenaline hydrochloride		β adrenergic receptor	99.86%
Norepinephrine	α1-adrenergic receptor α2-adrenergic receptor	Beta-1 adrenergic receptor	99.61%
Propranolol hydrochloride		β adrenergic receptor	99.95%
Propranolol		β adrenergic receptor	99.91%
Phenylephrine	α adrenergic receptor		99.98%
Agmatine	α2-adrenergic receptor
KMCA-0011	Alpha-2C adrenergic receptor, Ki: 56.7 nM		99.88%
D-Mannitol		Beta-3 adrenergic receptor	99.93%
Zenidolol hydrochloride		β adrenergic receptor	99.74%
CL 316243		β adrenergic receptor	99.98%
Norepinephrine hydrochloride	α1-adrenergic receptor α2-adrenergic receptor	Beta-1 adrenergic receptor	99.95%
Atenolol		Beta-1 adrenergic receptor, Ki: 697 nM	98.85%
Metoprolol		β1 adrenoceptor	99.99%
Phenylephrine hydrochloride	α adrenergic receptor		99.99%
Clozapine	α2-adrenergic receptor, Ki: 51 nM (Inhibitor)		99.84%
Dexmedetomidine	α2-adrenergic receptor, Ki: 1.08 nM		99.93%
Prazosin hydrochloride	α adrenergic receptor		99.89%
Dexmedetomidine hydrochloride	α2-adrenergic receptor, IC₅₀: 1.08 nM		99.94%
Nadolol		β adrenergic receptor	99.98%
Salbutamol		β adrenergic receptor	99.53%
Norepinephrine bitartrate monohydrate	α1-adrenergic receptor α2-adrenergic receptor	Beta-1 adrenergic receptor	99.96%
Mirabegron		β adrenergic receptor	99.90%
SR59230A		β adrenergic receptor	98.0%
(S)-Timolol maleate		β adrenergic receptor	99.80%
Salmeterol		β2 adrenoceptor, pEC₅₀: 9.6 β1 adrenoceptor, pEC₅₀: 6.1 β3 adrenoceptor, pEC₅₀: 5.9	99.69%
Labetalol	α1-adrenergic receptor	β-adrenoceptor	99.94%
Phentolamine	α1-adrenergic receptor α2-adrenergic receptor		99.94%
Dobutamine hydrochloride	α adrenergic receptor	β adrenergic receptor	99.60%
Formoterol fumarate		β2 adrenoceptor	99.95%
Phenylacetylglycine		β2 adrenoceptor	99.42%
Atipamezole	α adrenergic receptor		99.84%
Guanfacine hydrochloride	α adrenergic receptor		99.98%
Clonidine hydrochloride	α adrenergic receptor		99.94%
Mirtazapine	α2-adrenergic receptor, pKi: 6.95		99.94%
Tamsulosin	α1-adrenergic receptor		99.80%
Atipamezole hydrochloride	α adrenergic receptor		99.97%
L748337		Beta-3 adrenergic receptor, Ki: 4 nM Beta-2 adrenergic receptor, Ki: 204 nM Beta-1 adrenergic receptor, Ki: 390 nM	99.0%
Octopamine hydrochloride	α2-adrenergic receptor		99.90%
Metoprolol tartrate		β1 adrenoceptor	99.98%
Higenamine		β adrenergic receptor	99.31%
Methyldopa	α adrenergic receptor		99.87%
Vilanterol trifenatate		β adrenergic receptor	99.82%
Paliperidone	α adrenergic receptor		99.43%
Terbutaline		Beta-2 adrenergic receptor	99.94%
Terazosin hydrochloride	α adrenergic receptor		99.90%
Acebutolol hydrochloride		β1 adrenoceptor	99.70%
Metoprolol succinate		β1 adrenoceptor	99.56%
Bufuralol		β-adrenoceptor	99.25%
Salbutamol hemisulfate		β adrenergic receptor	98.0%
Harmane	α2-adrenergic receptor, IC₅₀: 18 μM		99.91%
Olodaterol		β2 adrenoceptor, EC₅₀: 0.1 nM	99.85%
Bisoprolol hemifumarate		Beta-1 adrenergic receptor	99.84%
Medetomidine hydrochloride	α2-adrenergic receptor, Ki: 1.08 nM α1-adrenergic receptor, Ki: 1750 nM		99.87%
Bufuralol hydrochloride		β adrenergic receptor	≥99.0%
Fenoterol hydrobromide		β adrenergic receptor	99.97%
Butaxamine hydrochloride		Beta-2 adrenergic receptor	99.87%
Brimonidine tartrate	α adrenergic receptor		99.68%
Carazolol		β1 adrenoceptor β2 adrenoceptor β3 adrenoceptor	99.78%
Phentolamine mesylate	α adrenergic receptor		99.90%
Blonanserin	α2-adrenergic receptor, Ki: 530 (Rat c nM α1-adrenergic receptor, Ki: 26.7 (Rat nM		99.91%
Bisoprolol		Beta-1 adrenergic receptor	99.78%
Vibegron		β3 adrenoceptor, EC₅₀: 1.1 nM	98.09%
SR59230A hydrochloride		β adrenergic receptor	99.81%
Indacaterol		β adrenergic receptor	99.98%
Norepinephrine tartrate	α1-adrenergic receptor α2-adrenergic receptor	Beta-1 adrenergic receptor	99.96%
Brimonidine	α adrenergic receptor		99.98%
Fenoterol		β adrenergic receptor	99.08%
(S)-(-)-Propranolol hydrochloride		β adrenergic receptor	99.97%
BMY 7378	rat α_1A-adrenergic receptor, Ki: 800 nM hamster alpha_1B-adrenergic receptor, Ki: 600 nM rat alpha_1D-adrenergic receptor, Ki: 2 nM		99.92%
Ecopipam hydrochloride	Alpha-2A adrenergic receptor, Ki: 731 nM		99.46%
Doxazosin mesylate	α adrenergic receptor		98.49%
Tamsulosin hydrochloride	α1-adrenergic receptor		99.76%
Salmeterol xinafoate		β2 adrenoceptor, pEC₅₀: 9.6 β1 adrenoceptor, pEC₅₀: 6.1 β3 adrenoceptor, pEC₅₀: 5.9	99.88%
Reboxetine mesylate	α adrenergic receptor		99.71%
Phentolamine hydrochloride	α1-adrenergic receptor α2-adrenergic receptor		99.91%
Terbutaline sulfate		β adrenergic receptor	99.95%
Vilanterol		β adrenergic receptor	99.30%
Guanfacine	α adrenergic receptor		99.85%
Dobutamine	α adrenergic receptor	β adrenergic receptor	98.75%
Synephrine		β adrenergic receptor	98.0%
(R)-Carvedilol		β adrenergic receptor	98.78%
Oxprenolol hydrochloride		β-adrenoceptor, Ki: 7.1 nM	99.86%
Metaproterenol hemisulfate		β adrenergic receptor	99.44%
Xamoterol hemifumarate		β1 adrenoceptor	≥99.0%
Terazosin hydrochloride dihydrate	α adrenergic receptor		99.92%
A-61603	α1A-adrenergic receptor		99.34%
Olodaterol hydrochloride		β2 adrenoceptor, EC₅₀: .1 nM	99.70%
Indacaterol maleate		β adrenergic receptor	99.82%
Esmolol hydrochloride		β-adrenoceptor	99.69%
Levonordefrin	α1-adrenergic receptor		98.62%
Pronethalol		β adrenergic receptor	99.88%
Penbutolol sulfate		β adrenergic receptor	98.89%
JP1302 dihydrochloride	human α2C-adrenoceptor, Ki: 28±2 nM human α2B-adrenoceptor, Ki: 1470±130 nM human α2A-adrenoceptor, Ki: 3150±50 nM rodent α2D-adrenoceptor, Ki: 1700±200 nM		99.94%
(R)-Propranolol hydrochloride		β adrenergic receptor	99.32%
LY 344864	rat α1-adrenergic receptor, Ki: 5.06 μM rat α2-adrenergic receptor, Ki: 3.69 μM		98.59%
Nefazodone hydrochloride	α1-adrenergic receptor		99.94%
Lubabegron		β adrenergic receptor	98.40%
Medetomidine	α2-adrenergic receptor, Ki: 1.08 nM α1-adrenergic receptor, Ki: 1750 nM		99.97%
Talipexole dihydrochloride	α2-adrenergic receptor, IC₅₀: 25 nM		99.80%
Zinterol hydrochloride		β adrenergic receptor	99.72%
Piribedil	α adrenergic receptor		99.92%
Isoetharine mesylate		β adrenergic receptor	99.05%
Nicergoline	α adrenergic receptor		99.31%
CGP 20712 A		β adrenergic receptor	99.0%
Ajmalicine	α1-adrenergic receptor α2-adrenergic receptor		99.23%
Ritodrine hydrochloride		β adrenergic receptor	99.81%
Asenapine	Alpha-2A adrenergic receptor, pKi: 8.9 Alpha-2C adrenergic receptor, pKi: 8.9 α1-adrenergic receptor, pKi: 8.9 Alpha-2B adrenergic receptor, pKi: 9.5		99.62%
Idazoxan hydrochloride	α adrenergic receptor		99.87%
Setiptiline	α adrenergic receptor		98.03%
Desglymidodrine	α1A-adrenergic receptor, pKi: 5.89 α1B-adrenergic receptor, pKi: 5.16 rat alpha_1D-adrenergic receptor, pKi: 5.78 human α2A-adrenoceptor, pKi: 5.83
Terazosin	α adrenergic receptor		99.28%
Tasipimidine sulfate	human α2A-adrenoceptor, pEC₅₀: 7.57 rat α2-adrenergic receptor, EC₅₀: 5.7 nM		99.32%
Indoramin	α adrenergic receptor		99.03%
Naftopidil	Alpha-1A adrenergic receptor, Ki: 3.7 nM Alpha-1B adrenergic receptor, Ki: 20 nM Alpha-1D adrenergic receptor, Ki: 1.2 nM		98.14%
Atenolol (Standard)		Beta-1 adrenergic receptor
Talinolol		Beta-1 adrenergic receptor	99.64%
Alfuzosin	α adrenergic receptor		99.86%
Reproterol		β2 adrenoceptor	98.94%
Efaroxan hydrochloride	α adrenergic receptor		99.80%
Midodrine hydrochloride	α adrenergic receptor		99.9%
Levalbuterol hydrochloride		β adrenergic receptor	99.58%
Clozapine (Standard)	α2-adrenergic receptor
Zotepine	α adrenergic receptor		99.80%
Xylometazoline hydrochloride	Alpha-1A adrenergic receptor, Ki: 0.05 μM Alpha-1B adrenergic receptor, Ki: 0.30 μM Alpha-1D adrenergic receptor, Ki: 0.15 μM Alpha-2A adrenergic receptor, Ki: 0.88 μM Alpha-2B adrenergic receptor, Ki: 1.7 μM Alpha-2C adrenergic receptor, Ki: 0.19 μM		99.94%
Levobunolol hydrochloride		β adrenergic receptor	99.95%
Metoprolol-d₇ hydrochloride		β adrenergic receptor	99.71%
NP10679	Alpha-1A adrenergic receptor, IC₅₀: 0.154 μM Alpha-1A adrenergic receptor, Ki: 0.603 μM Alpha-1B adrenergic receptor, Ki: 1.92 μM Alpha-1D adrenergic receptor, Ki: 0.495 μM Alpha-2C adrenergic receptor, Ki: 3.09 μM		98.40%
Vatinoxan hydrochloride	α adrenergic receptor		99.79%
Tulobuterol		β adrenergic receptor	99.69%
Denopamine		β adrenergic receptor	98.29%
Tizanidine	α adrenergic receptor		99.58%
Arformoterol tartrate		Beta-2 adrenergic receptor, Kd: 2.9 nM	99.63%
BODIPY FL prazosin	α1A-adrenergic receptor, Ki: 14.5 nM α1B-adrenergic receptor, Ki: 43.3 nM		99.71%
Lofexidine	α adrenergic receptor		99.08%
Celiprolol hydrochloride		β adrenergic receptor, Ki: 0.14-8.3 μM	99.98%
Metipranolol		β1 adrenoceptor, pA2: 8.3 β2 adrenoceptor, pA2: 8.4	98.15%
Midodrine	α adrenergic receptor		99.67%
(S,S)-BRL-37344 sodium		β adrenergic receptor	99.90%
Tizanidine hydrochloride	α adrenergic receptor		99.93%
Ecopipam	Alpha-2A adrenergic receptor, Ki: 731 nM		99.77%
Landiolol hydrochloride		Beta-1 adrenergic receptor	99.96%
BMS-466442	α adrenergic receptor, IC₅₀: ≥10 μM		98.0%
Methyldopa hydrate	α adrenergic receptor		99.95%
(+)-Penbutolol		β adrenergic receptor
Etilefrine hydrochloride	α1-adrenergic receptor	Beta-1 adrenergic receptor	99.90%
LM-189 free base		β2 adrenoceptor	99.70%
Gallamine Triethiodide		β-adrenoceptor	99.56%
Lofexidine hydrochloride	α adrenergic receptor		99.72%
Practolol		β adrenergic receptor	99.80%
CGP 12177 hydrochloride		Beta-1 adrenergic receptor, Ki: 0.9 nM Beta-2 adrenergic receptor, Ki: 4 nM Beta-3 adrenergic receptor, Ki: 88 nM	99.69%
Protokylol hydrochloride		Beta-2 adrenergic receptor	99.07%
Propranolol-d₇ hydrochloride		β adrenergic receptor	98.47%
Clorprenaline hydrochloride		β adrenergic receptor	99.90%
Methyldopate	α adrenergic receptor
Bevantolol hydrochloride	α adrenergic receptor	β adrenergic receptor	98.98%
Melperone	α2-adrenergic receptor, Kd: 150 nM α1-adrenergic receptor, Kd: 180 nM		99.84%
Cyanopindolol		β3 adrenoceptor	99.24%
Apraclonidine hydrochloride	α adrenergic receptor		98.96%
Dopexamine hydrochloride		β adrenergic receptor	98.04%
(R)-(+)-Atenolol		β adrenergic receptor	≥99.0%
Timolol		β adrenergic receptor
Ulimorelin	α adrenergic receptor
Salmeterol-d₃		β adrenergic receptor	98.04%
4-Hydroxypropranolol hydrochloride		β adrenergic receptor	99.73%
Spiroxatrine	α2-adrenergic receptor		99.25%
Dapiprazole hydrochloride	α1-adrenergic receptor		99.26%
Dicentrine	α adrenergic receptor		99.94%
Cimaterol		β-adrenoceptor	99.13%
LY377604		β adrenergic receptor	99.54%
Amibegron hydrochloride		β adrenergic receptor	≥99.0%
Hexoprenaline		β-adrenoceptor
Terbutaline sulfate (Standard)		β adrenergic receptor
AVN-101 hydrochloride	Alpha-1D adrenergic receptor, Ki: 30.2 nM Alpha-1B adrenergic receptor, Ki: 9.4 nM Alpha-2A adrenergic receptor, Ki: 1.77 nM Alpha-2C adrenergic receptor, Ki: 3.55 nM Alpha-1A adrenergic receptor, Ki: 18.9 nM Alpha-2B adrenergic receptor, Ki: 0.41 nM		99.59%
Solabegron		β adrenergic receptor	99.89%
Urapidil hydrochloride	α1-adrenergic receptor, pIC₅₀: 6.13 α2-adrenergic receptor, pIC₅₀: 4.38		99.86%
Harmane hydrochloride	α2-adrenergic receptor, IC₅₀: 18 μM		99.88%
Alfuzosin hydrochloride	α adrenergic receptor		99.72%
Mabuterol		Beta-2 adrenergic receptor	99.96%
Abanoquil	α1-adrenergic receptor		98.07%
(S)-Terazosin	α adrenergic receptor		99.71%
HOKU-81		Beta-2 adrenergic receptor
Prenalterol		β1 adrenoceptor	99.18%
Detomidine hydrochloride	α adrenergic receptor		99.83%
Arformoterol		Beta-2 adrenergic receptor, Kd: 2.9 nM	99.96%
Clozapine hydrochloride	α2-adrenergic receptor, Ki: 51 nM		99.83%
MT-1207	α1D-adrenergic receptor, IC₅₀: 0.086 nM α1D-adrenergic receptor, Ki: 0.69 nM α1B-adrenergic receptor, IC₅₀: 0.15 nM α1B-adrenergic receptor, Ki: 1.40 nM α1A-adrenergic receptor, IC₅₀: 0.1 nM		99.96%
Mibenratide		Beta-1 adrenergic receptor	99.47%
Nifenalol hydrochloride		β-adrenoceptor	99.93%
Amidephrine	α1-adrenergic receptor
(+)-Niguldipine hydrochloride	α1-adrenergic receptor, Ki: 78 nM		98.06%
ST91	α2-adrenergic receptor		99.75%
AP-7-168		Beta-2 adrenergic receptor	99.89%
Butyryltimolol		β adrenergic receptor	98.0%
JP1302	human α2C-adrenoceptor, Ki: 28±2 nM human α2B-adrenoceptor, Ki: 1470±130 nM human α2A-adrenoceptor, Ki: 3150±50 nM rodent α2D-adrenoceptor, Ki: 1700±200 nM		98.68%
Acebutolol		β1 adrenoceptor	99.70%
DL 071IT		β adrenergic receptor	98.81%
BMY 14802	α1-adrenergic receptor		98.07%
α1A-AR Degrader 9c	α1A-adrenergic receptor, DC₅₀: 2.86 μM
Mirtazapine (Standard)	α2-adrenergic receptor
(+)-Sotalol		β-adrenoceptor	99.89%
Carpipramine	α1-adrenergic receptor α2-adrenergic receptor
Ro 363 hydrochloride		β adrenergic receptor
Synephrine hydrochloride		β adrenergic receptor	99.66%
Undecylenoyl phenylalanine		β-adrenoceptor
Etoperidone	α1-adrenergic receptor, Kd: 38 nM α2-adrenergic receptor, Kd: 570 nM
BMY-14802 hydrochloride	α1-adrenergic receptor		98.02%
LM-189		β2 adrenoceptor, Ki: 0.063 nM Beta-1 adrenergic receptor, Ki: 28 nM
ARC 239 dihydrochloride	Alpha-2B adrenergic receptor		99.20%
MK-761 free base		Beta-2 adrenergic receptor	99.56%
CL 316243 free acid		β3 adrenoceptor	99.37%
4-Hydroxypropranolol-d₇ hydrochloride		β adrenergic receptor	98.68%
Buflomedil hydrochloride	rat α_1A-adrenergic receptor, Ki: 4.06 μM α1B-adrenergic receptor, Ki: 6.84 μM		99.81%
Ecopipam hydrobromide	Alpha-2A adrenergic receptor, Ki: 731 nM		99.0%
ORM-10921 free base	Alpha-2C adrenergic receptor, Ki: 1.4 nM		98.08%
Brombuterol-d₉		β adrenergic receptor	99.0%
Nadolol-d₉		β adrenergic receptor
Clorprenaline		β adrenergic receptor	99.33%
RS-79948-197	rat α2A receptor, Kd: 0.42 nM rat α2B recepter, Kd: 0.18 nM rat α2C recepter, Kd: 0.19 nM human α2A-adrenoceptor, Kd: 0.6 nM human α2B-adrenoceptor, Kd: 0.46 nM human α2C-adrenoceptor, Kd: 0.77 nM		99.5%
Prazobind	Alpha-1A adrenergic receptor, IC₅₀: 1 nM Alpha-1B adrenergic receptor, IC₅₀: 1 nM
Bunazosin	α1-adrenergic receptor		98.52%
Iloperidone carboxylic acid	human α2C-adrenoceptor, pKi: 7.32 human α2A-adrenoceptor, pKi: 6.42 rat α1-adrenergic receptor, pKi: 7.67 human α2B-adrenoceptor, pKi: 7.08		99.6%
Fluparoxan	α2-adrenergic receptor		99.66%
Metaterol		β adrenergic receptor
Amosulalol	α1-adrenergic receptor	Beta-1 adrenergic receptor	98.69%
p-F-HHSiD hydrochloride	α1-adrenergic receptor		99.0%
Diacetolol-d₇		β adrenergic receptor	99.9%
GS-5759		β2 adrenoceptor	99.21%
Bupranolol		β-adrenoceptor	98.90%
Levalbuterol		β adrenergic receptor
Benzquinamide hydrochloride	Alpha-2A adrenergic receptor Alpha-2B adrenergic receptor Alpha-2C adrenergic receptor		99.14%
Napamezole hydrochloride	α2-adrenergic receptor, Ki: 28 nM α1-adrenergic receptor, Ki: 93 nM		98.97%
Bunitrolol		β-adrenoceptor	99.79%
Xamoterol		β1 adrenoceptor
(RS)-Butyryltimolol		β adrenergic receptor	98.0%
α2A-AR agonist 1	Alpha-2A adrenergic receptor, EC₅₀: 0.23 nM Alpha-1A adrenergic receptor, EC₅₀: 2.5 nM Alpha-2B adrenergic receptor, EC₅₀: 16.3 nM Alpha-2C adrenergic receptor, EC₅₀: 21.3 nM		99.92%
L-771688	α adrenergic receptor		99.46%
ARC 239	human α2C-adrenoceptor, pKi: 6.95 Alpha-2C adrenergic receptor, pKi: 7.06		99.71%
Midaglizole hydrochloride	α adrenergic receptor		99.67%
Nafetolol		Beta-1 adrenergic receptor	98.24%
Zinterol		β adrenergic receptor
ST1936	α2-adrenergic receptor, Ki: 300 nM (rat) α2-adrenergic receptor, Ki: 300 nM (human) α1-adrenergic receptor, Ki: 390 nM (rat)		98.66%
Oxyfedrine		β-adrenoceptor
AGN 192836	α adrenergic receptor		99.49%
(Rac)-Rotigotine hydrochloride	Alpha-2B adrenergic receptor		98.11%
Clenproperol		β adrenergic receptor	99.44%
Xylometazoline	Alpha-1A adrenergic receptor, Ki: 0.05 μM Alpha-1B adrenergic receptor, Ki: 0.30 μM Alpha-1D adrenergic receptor, Ki: 0.15 μM Alpha-2A adrenergic receptor, Ki: 0.88 μM Alpha-2B adrenergic receptor, Ki: 1.7 μM Alpha-2C adrenergic receptor, Ki: 0.19 μM
OPC-28326	α adrenergic receptor		99.46%
Mapenterol hydrochloride		β adrenergic receptor	99.56%
β2AR-IN-15		β2 adrenoceptor, Kd: 1.7 μM
Isoetharine		β adrenergic receptor
Timolol hemihydrate		β adrenergic receptor
Blonanserin dihydrochloride	α2-adrenergic receptor, Ki: 530 nM α1-adrenergic receptor, Ki: 26.7 nM
(R,R)-Reboxetine mesylate	α adrenergic receptor
Sotalol		β-adrenoceptor
AGN-190851	Alpha-2A adrenergic receptor
Dobutamine tartrate	α adrenergic receptor	β adrenergic receptor
Mivazerol	α2-adrenergic receptor
Scoulerine hydrochloride	Alpha-1D adrenergic receptor
Ritodrine		β adrenergic receptor
CAXII-IN-3		Beta-2 adrenergic receptor Beta-1 adrenergic receptor Beta-3 adrenergic receptor
Etoperidone hydrochloride	α1-adrenergic receptor, Kd: 38 nM α2-adrenergic receptor, Kd: 570 nM
Metoprolol fumarate		β1 adrenoceptor
Isamoltan hydrochloride		β-adrenoceptor, IC₅₀: 8.4 nM
Bopindolol fumarate		β1 adrenoceptor β2 adrenoceptor β3 adrenoceptor
Bunolol		β-adrenoceptor
(±)-WB 4101	α1-adrenergic receptor
Docarpamine	α adrenergic receptor
Trimazosin	α1-adrenergic receptor
Naftopidil dihydrochloride	Alpha-1A adrenergic receptor, Ki: 3.7 nM Alpha-1B adrenergic receptor, Ki: 20 nM Alpha-1D adrenergic receptor, Ki: 1.2
Flestolol sulfate		β adrenergic receptor
LY 78335	α2-adrenergic receptor, IC₅₀: 10 μM
2-(2-Methoxyphenoxy)ethylamine hydrochloride	α1-adrenergic receptor		99.65%
Rezatomidine	α2-adrenergic receptor
Fenoxazoline	α1-adrenergic receptor
β2AR antagonist 1		Beta-2 adrenergic receptor
Cloranolol		β-adrenoceptor
BRL 35135		β3 adrenoceptor
Levalbuterol hemitartrate		β adrenergic receptor	98.71%
Nipradolol	α1-adrenergic receptor
SGB-1534 hydrochloride	α1-adrenergic receptor
Piribedil dihydrochloride	α adrenergic receptor
Celiprolol		β adrenergic receptor, Ki: 0.14-8.3 μM
Metoprolol-d₆ tartrate		β adrenergic receptor
ent-Levobunolol hydrochloride		β adrenergic receptor
Zolertine hydrochloride	α1B-adrenergic receptor, pKi: 6.81 (in rat liver membrane) α1A-adrenergic receptor, pKi: 6.35 (in rabbit liver membrane)
DL-017	α1-adrenergic receptor
β-Blocker B-24/76		β adrenergic receptor
SB-206606		Beta-3 adrenergic receptor
α2AR agonist 1	α2-adrenergic receptor
Oxprenolol		β-adrenoceptor, Ki: 7.1 nM
(+)-Niguldipine	α1-adrenergic receptor, Ki: 52 pM
Bopindolol		β2 adrenoceptor Beta-1 adrenergic receptor Beta-3 adrenergic receptor
L-657743	α2-adrenergic receptor
Nifenalol		Beta-1 adrenergic receptor
α1A/1D-Adrenoceptor antagonist-1	α1A-adrenergic receptor, IC₅₀: 20.26 nM α1D-adrenergic receptor, IC₅₀: 164.9 nM α1B-adrenergic receptor, IC₅₀: 1912 nM α1A-adrenergic receptor, pA2: 7.68 α1D-adrenergic receptor, pA2: 8.67 α1B-adrenergic receptor, pA2: 6.55		99.65%
(S)-Trimetoquinol hydrochloride		β-adrenoceptor
Melperone hydrochloride	α2-adrenergic receptor, Kd: 150 nM α1-adrenergic receptor, Kd: 180 nM
Fipamezole	human α2A-adrenoceptor, Ki: 9.2 nM human α2B-adrenoceptor, Ki: 17 nM human α2C-adrenoceptor, Ki: 55 nM
(E)-Guanabenz	α adrenergic receptor
Tazolol		β-adrenoceptor
α2C adrenoceptor agonist 1	Alpha-2C adrenergic receptor, EC₅₀: 108 nM Alpha-2C adrenergic receptor, Ki: 12 nM
hERG-IN-3	α1A-adrenergic receptor, IC₅₀: 270 nM	Beta-2 adrenergic receptor, IC₅₀: 14 nM
Rec 15/2615 hydrochloride	α1A-adrenergic receptor, Ki: 1.9 nM α1B-adrenergic receptor, Ki: 0.3 nM Alpha-1D adrenergic receptor, Ki: 2.6 nM
Fenoterol hydrobromide (Standard)		β adrenergic receptor
Acebutolol-d₇		β adrenergic receptor
SL-89.0591	α1-adrenergic receptor
Isamoltane hemifumarate		β-adrenoceptor, IC₅₀: 8.4 nM
Isoprenaline hemisulfate		β adrenergic receptor	98.10%
S(-)-Bisoprolol fumarate		β adrenergic receptor
TAK-259 hydrochloride	Alpha-1D adrenergic receptor, Ki: 1.1 nM
Butaxamine		β2 adrenoceptor
KRG-3332 hydrochloride	α1A-adrenergic receptor
LAS190792		β2 adrenoceptor, pIC₅₀: 9.1 β3 adrenoceptor, pIC₅₀: 5.6 β1 adrenoceptor, pIC₅₀: 7.5
SM-11044		β1 adrenoceptor, Ki: 18.1 μM β2 adrenoceptor, Ki: 4.1 μM β3 adrenoceptor, Ki: 1.3 μM
CYD-1-79	Alpha-2A adrenergic receptor Alpha-2B adrenergic receptor
Ajmalicine hydrochloride	α1-adrenergic receptor α2-adrenergic receptor
S(-)-Bisoprolol		β adrenergic receptor
SM-2470	α adrenergic receptor
Rimiterol		Beta-2 adrenergic receptor
Bisoprolol fumarate		Beta-1 adrenergic receptor
Tracizoline	α2-adrenergic receptor
Procaterol		β2 adrenoceptor
Enciprazine dihydrochloride	α1-adrenergic receptor
β2AR/M3-receptor agonist-1		β2 adrenoceptor, pEC₅₀: >9.2
(±)-Desisopropylpropranolol		β adrenergic receptor
(S)-Bopindolol		β-adrenoceptor
BRL-41992	Alpha-2A adrenergic receptor, Ki: 1.1 nM Alpha-2B adrenergic receptor, Ki: 103.3 nM
CGP 12177		Beta-1 adrenergic receptor, Ki: 0.9 nM Beta-2 adrenergic receptor, Ki: 4 nM Beta-3 adrenergic receptor, Ki: 88 nM
(±)-Penbutolol		Beta-1 adrenergic receptor
RWJ52353	Alpha-2D adrenergic receptor, Ki: 1.5 nM Alpha-2A adrenergic receptor, Ki: 254 nM α1-adrenergic receptor, Ki: 443 nM Alpha-2B adrenergic receptor, Ki: 621 nM
Mazapertine	α1-adrenergic receptor, Ki: 1.3 nM
Naftopidil hydrochloride	Alpha-1A adrenergic receptor, Ki: 3.7 nM Alpha-1B adrenergic receptor, Ki: 20 nM Alpha-1D adrenergic receptor, Ki: 1.2 nM
Harmane (Standard)	α2-adrenergic receptor
Ro 70‐0004	Alpha-1A adrenergic receptor, pKi: 8.9
NLX-219	α1-adrenergic receptor, pKi: 6.29
VUF26034		Beta-2 adrenergic receptor
Meluadrine		β2 adrenoceptor
ST1936 oxalate	α2-adrenergic receptor, Ki: 300 nM (rat) α2-adrenergic receptor, Ki: 300 nM (human) α1-adrenergic receptor, Ki: 390 nM (rat)
Meluadrine tartrate		β2 adrenoceptor
Cimbuterol-d₉		β adrenergic receptor
Z8779877149	α2-adrenergic receptor, Ki: 180 nM α2-adrenergic receptor, EC₅₀: 440 nM
Salbutamol adipate		β adrenergic receptor
NRA-0562	α1-adrenergic receptor
Azapetine	rat α1-adrenergic receptor, IC₅₀: 0.205 μM rat α2-adrenergic receptor, IC₅₀: 1.3 μM
ICI 147798		β-adrenoceptor, pkB: 8.8
SUN-1334H free base	Alpha-1D adrenergic receptor, IC₅₀: 7.76 μM
Clencyclohexerol		β2 adrenoceptor
TAK-259	Alpha-1D adrenergic receptor, Ki: 1.1 nM
Dapiprazole	α1-adrenergic receptor
Apraclonidine	α adrenergic receptor
Etilefrine hydrochloride (Standard)	α1-adrenergic receptor	Beta-1 adrenergic receptor
CACPD2011a-0001278239		Beta-2 adrenergic receptor
Phenylethanolamine A-d₃		β adrenergic receptor
Moprolol		Beta-1 adrenergic receptor
CP-114271		β3 adrenoceptor
Pronethalol hydrochloride		β adrenergic receptor
N-5984		β-adrenoceptor
Asenapine citrate	Alpha-2A adrenergic receptor, pKi: 8.9 Alpha-2C adrenergic receptor, pKi: 8.9 α1-adrenergic receptor, pKi: 8.9 Alpha-2B adrenergic receptor, pKi: 9.5
L742791		Beta-3 adrenergic receptor
Delequamine hydrochloride	α2-adrenergic receptor, pKi: 9.5 α1-adrenergic receptor, pKi: 5.3
Metaproterenol		β adrenergic receptor
CSP-2503	α1-adrenergic receptor, Ki: >1000 nM
Clenproperol-d₇		β adrenergic receptor
SNAP-6201	α1A-adrenergic receptor, Ki: 0.2 nM α1B-adrenergic receptor, Ki: 260 nM α1D-adrenergic receptor, Ki: 350 nM rat α_1A-adrenergic receptor, Ki: 0.27 nM
(2S,3S)-Zenidolol hydrochloride		Beta-2 adrenergic receptor, pKi: 7.51 Beta-1 adrenergic receptor, pKi: 9.27
(±)-Penbutolol-d₉ hydrochloride		β adrenergic receptor
Dihydroergotamine	α adrenergic receptor
L-665871		β adrenergic receptor
Sibenadet		β2 adrenoceptor
Piperoxan	rat α1-adrenergic receptor, Ki: 360 nM
Fadolmidine hydrochloride	α2-adrenergic receptor
Levobunolol		β adrenergic receptor
Atiprosine	α1-adrenergic receptor, pA2: 8.11 α2-adrenergic receptor, pA2: 6.04
GSK-3β/G9a-IN-1	Alpha-2A adrenergic receptor
2-MPMDQ	α1-adrenergic receptor, Ki: 0.37 nM α2-adrenergic receptor, Ki: 1740 nM
Sulfinalol		β-adrenoceptor
Mabuterol-d₉		β adrenergic receptor
Pafenolol		Beta-1 adrenergic receptor
Agroclavine	α1-adrenergic receptor
Landiolol		Beta-1 adrenergic receptor
β2AR agonist 5		β2 adrenoceptor, EC₅₀: 0.19 nM
S(-)-Cyanopindolol hemifumarate		β3 adrenoceptor
Jingsongling	α1-adrenergic receptor α2-adrenergic receptor
Clozapine dihydrochloride	α2-adrenergic receptor, Ki: 51 nM
Zolertine	α1A-adrenergic receptor, pKi: 6.35 α1B-adrenergic receptor, pKi: 6.81
Terazosin-md	α1-adrenergic receptor
Pacrinolol		Beta-1 adrenergic receptor
GG-818	Alpha-1A adrenergic receptor, pKi: 9.7 Alpha-1B adrenergic receptor, pKi: 7.8 Alpha-1D adrenergic receptor, pKi: 7.6
A 131701	α1A-adrenergic receptor, Ki: 0.22 nM
SAR-150640		β3 adrenoceptor
Buflomedil	rat α_1A-adrenergic receptor, Ki: 4.06 μM α1B-adrenergic receptor, Ki: 6.84 μM
Fadolmidine	α2-adrenergic receptor
Methyldopate hydrochloride	α adrenergic receptor
Fadaltran	Alpha-2C adrenergic receptor
IP-66	α1-adrenergic receptor
LY 344864 hydrochloride	rat α1-adrenergic receptor, Ki: 5.06 μM rat α2-adrenergic receptor, Ki: 3.69 μM
BMS-201620		β3 adrenoceptor, Ki: 93 nM
AH 11110A	α1B-adrenergic receptor
Platelet aggregation-IN-3	α2-adrenergic receptor
Ractopamine		pig β₁AR, Kd: ~25 nM pig β₂AR, Kd: ~25 nM
BRL-37344		β3 adrenoceptor, EC₅₀: 5.3 nM β2 adrenoceptor, EC₅₀: 18 nM β1 adrenoceptor, EC₅₀: 570 nM
β2AR agonist /M-receptor antagonist-1		Beta-2 adrenergic receptor
Brombuterol-d₉ hydrochloride		β adrenergic receptor
CHF-6550		β2 adrenoceptor, pKi: 10.6
Arrestin-3 modulator-1		Beta-2 adrenergic receptor
Tasipimidine	human α2A-adrenoceptor, pEC₅₀: 7.57 rat α2-adrenergic receptor, EC₅₀: 5.7 nM
Metrenperone	α1-adrenergic receptor α2-adrenergic receptor
p-F-HHSiD	α1-adrenergic receptor
Zilpaterol-d₇		β adrenergic receptor
Bevantolol		Beta-1 adrenergic receptor
Doxazosin-d₈	α adrenergic receptor
ICI-170777		β adrenergic receptor
Photoazolol-1		β-adrenoceptor
TAAR1 agonist 3	Alpha-2A adrenergic receptor, pEC₅₀: 6
Fasobegron		β3 adrenoceptor, EC₅₀: 4.8 nM β1 adrenoceptor, EC₅₀: 250 nM
Levobetaxolol		β1 adrenoceptor, IC₅₀: 33.2 nM β2 adrenoceptor, IC₅₀: 2970 nM β3 adrenoceptor, IC₅₀: 709 nM
Todralazine		β adrenergic receptor
Methyl maslinate		β adrenergic receptor	98.0%
Arformoterol maleate		Beta-2 adrenergic receptor, Kd: 2.9 nM
A 80426 mesylate	α2-adrenergic receptor
Landiolol hydrochloride (Standard)		Beta-1 adrenergic receptor
Indacaterol xinafoate		β2 adrenoceptor
Mabuterol hydrochloride		Beta-2 adrenergic receptor
Fiduxosin hydrochloride	α1A-adrenergic receptor, IC₅₀: 0.16 nM α1B-adrenergic receptor, IC₅₀: 24.9 nM α1D-adrenergic receptor, IC₅₀: 0.92 nM
Bunitrolol hydrochloride		β-adrenoceptor
PF-9404C		β adrenergic receptor
Melperone (Standard)	α2-adrenergic receptor, Kd: 150 nM α1-adrenergic receptor, Kd: 180 nM
Sulfinalol hydrochloride		β-adrenoceptor
Melperone-d₄ hydrochloride	α2-adrenergic receptor, Kd: 150 nM α1-adrenergic receptor, Kd: 180 nM		99.84%
Xibenolol hydrochloride		β-adrenoceptor
SB251023		Beta-3 adrenergic receptor
Methyldopa hydrochloride	α adrenergic receptor
CHIR-2279	α1-adrenergic receptor, Ki: 5 nM
Hexoprenaline sulfate		β-adrenoceptor
RU 52583	α2-adrenergic receptor
Nemazoline	α1-adrenergic receptor α2-adrenergic receptor
Xamoterol hemifumarate (Standard)		β1 adrenoceptor
Org 6906	α2-adrenergic receptor, pKi: 6.5
Carbuterol hydrochloride		Beta-2 adrenergic receptor
α1A Adrenoceptor antagonist-1	α1A-adrenergic receptor, Ki: <20 nM
Clorprenaline-d₇		β adrenergic receptor
R 47 243	α2-adrenergic receptor
Esmolol		β adrenergic receptor
L-748328		β3 adrenoceptor, Ki: 3.7 nM
(rac)-Nebivolol-d₄		β adrenergic receptor
Cicloprolol hydrochloride		β adrenergic receptor
Pargolol hydrochloride		β adrenergic receptor
TD-5471 hydrochloride		β adrenergic receptor
Ko-3290		β adrenergic receptor
Delequamine	α2-adrenergic receptor, pKi: 9.5 α1-adrenergic receptor, pKi: 5.3
L-770644		Beta-3 adrenergic receptor, EC₅₀: 13 nM
SNAP8719 free base	Alpha-1D adrenergic receptor, pKi: 8.89 Alpha-2A adrenergic receptor, pKi: <5.0
Azepexole dihydrochloride	α adrenergic receptor
Buflomedil hydrochloride (Standard)	rat α_1A-adrenergic receptor, Ki: 4.06 μM α1B-adrenergic receptor, Ki: 6.84 μM
Ridazolol		Beta-1 adrenergic receptor
Trimazosin hydrochloride hydrate	α1-adrenergic receptor
Benzquinamide	α adrenergic receptor
QF0301B	α adrenergic receptor
α1 adrenoceptor-MO-1	α adrenergic receptor
Epanolol		β adrenergic receptor
Fenmetozole Tosylate	α adrenergic receptor
AR-08	α adrenergic receptor

Name
Email *

	Sorry, but the email address you supplied was invalid.